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Cis-22a

Cis-22a is a TRPV6 inhibitor (IC50 = 0.32 μM), which exhibits selectivity against related TRPV channels and calcium channels. cis-22a displays antiproliferative effects on T47D human breast cancer cells.

Product Specifications

CAS Number

1819366-84-1

Stability

≥ 2 years

Purity

>98% (HPLC)

Weight

449.51

Molecular Formula

C24H30F3N3O2

Notes

Research use only, not for human use.

Receptor

Calcium Channel | TRP/TRPV Channel

Available Sizes

Frequently Asked Questions

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