Cis-22a
Cis-22a is a TRPV6 inhibitor (IC50 = 0.32 μM), which exhibits selectivity against related TRPV channels and calcium channels. cis-22a displays antiproliferative effects on T47D human breast cancer cells.
Product Specifications
CAS Number
1819366-84-1
Stability
≥ 2 years
Purity
>98% (HPLC)
Weight
449.51
Molecular Formula
C24H30F3N3O2
Notes
Research use only, not for human use.
Receptor
Calcium Channel | TRP/TRPV Channel
Available Sizes
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