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NCGC00029283

NCGC00029283 is a potent inhibitor of Werner syndrome helicase-nuclease (WRN), displaying inhibitory activity against WRN helicase with an IC 50 value of 2.3 μM. Additionally, it exhibits inhibitory effects on Bloom syndrome protein helicase (BLM) and Fanconi anemia group J protein helicase (FANCJ) with IC 50 values of 12.5 μM and 3.4 μM, respectively.

Product Specifications

CAS Number

714240-31-0

Stability

≥ 2 years

Purity

>98% (HPLC)

Weight

337.3

Molecular Formula

C18H12FN3O3

Notes

Research use only, not for human use.

Receptor

DNA/RNA Synthesis

Available Sizes

Curated Selection

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