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Patamostat mesylate

Patamostat mesylate (E-3123) is a potent protease inhibitor with IC50 values of 39 nM for trypsin, 950 nM for plasmin, and 1.9 μM for thrombin. This compound demonstrates promising potential in suppressing the pathogenesis and development of acute pancreatitis.

Product Specifications

CAS Number

114568-32-0

Stability

≥ 2 years

Purity

>98% (HPLC)

Weight

508.57

Molecular Formula

C21H24N4O7S2

Notes

Research use only, not for human use.

Receptor

HDAC | Apoptosis

Available Sizes

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