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CB2R PAM

CB2R PAM is an orally active cannabinoid type 2 receptor (CB2Rs) positive allosteric modulator that enhances CP 55940 and 2-Arachidonylglycerol-stimulated [35S]GTPγS binding to CB2 receptors without affecting receptor activity in the absence of agonists. CB2R PAM shows anti-injury activity in a mouse model of neuropathic pain.

Product Specifications

CAS Number

2244579-87-9

Stability

≥ 2 years

Purity

>98% (HPLC)

Weight

435.33

Molecular Formula

C21H24BrFN2O2

Notes

Research use only, not for human use.

Receptor

Cannabinoid Receptor

Available Sizes

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