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Valiglurax

Valiglurax (VU2957), also known as VU0652957 and VU2957, is a potent, selective, CNS penetrant, and orally bioavailable mGlu4 PAM. VU2957 possessed attractive in vitro and in vivo pharmacological and DMPK properties across species. VU2957 was evaluated as a preclinical development candidate for the treatment of Parkinson’s disease.

Product Specifications

CAS Number

1976050-09-5

Stability

≥ 2 years

Purity

>98% (HPLC)

Weight

329.28

Molecular Formula

C16H10F3N5

Notes

Research use only, not for human use.

Receptor

GluR

Available Sizes

Curated Selection

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