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CCG-257081

CCG-257081 (MRTF/SRF-IN-1) is an inhibitor of cardiac myosin-related transcription factor and serum response factor (MRTF/SRF) that acts by inhibiting the Rho/MRTF/SRF pathway.CCG-257081 has shown efficacy in preventing bleomycin-induced fibrosis in several mouse models. CCG-257081 can be used in cancer prevention and fibrosis research.

Product Specifications

CAS Number

1922098-90-5

Stability

≥ 2 years

Purity

>98% (HPLC)

Weight

473.87

Molecular Formula

C24H19ClF3N3O2

Notes

Research use only, not for human use.

Receptor

Rho | Ras

Available Sizes

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