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Ponatinib Hydrochloride

Ponatinib Hydrochloride (AP-24534 Hydrochloride) is a hydrochloride of ponatinib. Ponatinib is an orally active multi-targeted kinase inhibitor with IC50s of 0.37 nM, 1.1 nM, 1.5 nM, 2.2 nM, and 5.4 nM for Abl, PDGFRα, VEGFR2, FGFR1, and Src, respectively.

Product Specifications

CAS Number

1114544-31-8

Stability

≥ 2 years

Purity

>98% (HPLC)

Weight

569.02

Molecular Formula

C29H28ClF3N6O

Notes

Research use only, not for human use.

Receptor

Src | PDGFR | VEGFR | FGFR

Available Sizes

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