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MNI 137

MNI 137 is a negative allosteric modulator of mGlu2. MNI 137 inhibits glutamate-induced calcium mobilization with IC50s of 8.3 and 12.6 nM for human and rat.

Product Specifications

CAS Number

946619-21-2

Stability

≥ 2 years

Purity

>98% (HPLC)

Weight

341.16

Molecular Formula

C15H9BrN4O

Notes

Research use only, not for human use.

Receptor

GluR

Available Sizes

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