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ML289

ML289 (VU0463597) is a potent, selective, and CNS-penetrant negative allosteric modulator of mGlu3 (IC50=0.66 μM), with over 15-fold selectivity compared to mGlu2 and no activity against mGlu5.

Product Specifications

Stability

≥ 2 years

Purity

>98% (HPLC)

Weight

349.42

Molecular Formula

C22H23NO3

Notes

Research use only, not for human use.

Receptor

GluR

CAS Number

1382481-79-9

Available Sizes

Curated Selection

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