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Cyclapolin 9

Cyclapolin 9 is a selective, potent, and ATP-competitive inhibitor of polo-like kinase 1 (PLK1) with an IC50 of 500 nM, and has not shown activity against other kinases.

Product Specifications

CAS Number

40533-25-3

Stability

≥ 2 years

Purity

>98% (HPLC)

Weight

307.21

Molecular Formula

C9H4F3N3O4S

Notes

Research use only, not for human use.

Receptor

PLK

Available Sizes

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