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AG 045572

AG 045572 is a potent GnRH receptor antagonist that inhibits the GnRH receptor in humans and rats with Ki values of 6.0 nM and 3.8 nM, respectively.AG 045572 is metabolized by CYP3A and inhibits testosterone.

Product Specifications

Stability

≥ 2 years

Purity

>98% (HPLC)

Weight

491.62

Molecular Formula

C30H37NO5

Notes

Research use only, not for human use.

Receptor

P450 | GNRH Receptor

CAS Number

263847-55-8

Available Sizes

Curated Selection

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