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MG-115

MG-115 (Z-LL-Nva-CHO) is a potent and reversible inhibitor of proteasome , with K i s of 21 nM and 35 nM for 20S and 26S proteasome, respectively. MG-115 specifically inhibit the chymotrypsin-like activity of the proteasome, induces p53-dependent apoptosis .

Product Specifications

CAS Number

133407-86-0

Stability

≥ 2 years

Purity

>98% (HPLC)

Weight

461.59

Molecular Formula

C25H39N3O5

Notes

Research use only, not for human use.

Receptor

Proteasome

Available Sizes

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