PF-4981517
PF-4981517 (CYP3cide) is a efficient, specific and time-dependent inhibitor of cytochrome P4503A4 (CYP3A4) . The IC 50 values for CYP3A activity are 0.03 μM,17 μM, and 71 μM for CYP3A4, CYP3A5, and CYP3A7, respectively. PF-4981517 is able to be used to distinguish the contributions of CYP3A4 versus CYP3A5 on drug Metabolism.
Product Specifications
CAS Number
1390637-82-7
Stability
≥ 2 years
Purity
>98% (HPLC)
Weight
456.59
Molecular Formula
C26H32N8
Notes
Research use only, not for human use.
Receptor
P450
Available Sizes
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