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Tesaglitazar

Tesaglitazar is a potent and selective peroxide PPARα / γ receptor dual agonist with a more potent affinity for PPARγ than PPARα, The EC50 values for rat PPARα and human PPARα were 13.4 μM and 3.6 μM, respectively, and 0.2 μM for rat PPARγ and human PPARγ. Tesaglitazar induced DNA synthesis and fibrosarcoma formation in rat subcutaneous mesenchymal cells.

Product Specifications

Stability

≥ 2 years

Purity

>98% (HPLC)

Weight

408.47

Molecular Formula

C20H24O7S

Notes

Research use only, not for human use.

Receptor

PPAR

CAS Number

251565-85-2

Available Sizes

Curated Selection

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