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M77976

M77976 is a selective ATP-competitive inhibitor of pyruvate dehydrogenase kinase 4 (PDK4) with an inhibitory effect on PDK4, having an IC50 value of 648 μM. It is used for research related to obesity and diabetes.

Product Specifications

CAS Number

394237-61-7

Stability

≥ 2 years

Purity

>98% (HPLC)

Weight

296.32

Molecular Formula

C17H16N2O3

Notes

Research use only, not for human use.

Receptor

PDK

Available Sizes

Curated Selection

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