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TPN171

TPN171 is potent PDE5 inhibitor with subnanomolar potency for PDE5 and good selectivity over PDE6, which has the potential for the treatment of pulmonary arterial hypertension (PAH) . TPN171 was proven to exert a longer lasting effect than sildenafil in animal models, providing a foundation for a once-daily oral administration for its clinical use.

Product Specifications

CAS Number

1229018-87-4

Stability

≥ 2 years

Purity

>98% (HPLC)

Weight

441.57

Molecular Formula

C24H35N5O3

Notes

Research use only, not for human use.

Receptor

PDE

Available Sizes

Frequently Asked Questions

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