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TCMDC-135051

TCMDC-135051 is a potent and selective PfCLK3 protein kinase inhibitor demonstrating significant antiparasiticidal activity (EC50=320 nM) while exhibiting minimal off-target toxicity. It effectively hinders the transition from trophozoite to schizont, impairs transcription, and diminishes transmission to the mosquito vector.

Product Specifications

CAS Number

2413716-15-9

Stability

≥ 2 years

Purity

>98% (HPLC)

Weight

471.59

Molecular Formula

C29H33N3O3

Notes

Research use only, not for human use.

Receptor

Others

Available Sizes

Curated Selection

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