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Lusaperidone

Lusaperidone (R107474) is a potent α2-adrenergic receptor antagonist, a potential radioligand for the α (2) -adrenergic receptor, with inhibitory effects on α2A and α2C, with Ki values of 0.13 and 0.15 nM, respectively.

Product Specifications

CAS Number

214548-46-6

Stability

≥ 2 years

Purity

>98% (HPLC)

Weight

359.42

Molecular Formula

C22H21N3O2

Notes

Research use only, not for human use.

Receptor

Adrenergic Receptor

Available Sizes

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