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I-OMe-Tyrphostin AG 538

I-OMe-Tyrphostin AG 538 is a specific IGF-1R inhibitor and ATP-competitive inhibitor of PI5P4Kα (IC50: 1 µM) .I-OMe-Tyrphostin AG 538 inhibits IGF-1R-mediated signaling and exhibits preferential cytotoxicity to nutrient-deficient PANC1 cells.

Product Specifications

CAS Number

1094048-77-7

Stability

≥ 2 years

Purity

>98% (HPLC)

Weight

437.19

Molecular Formula

C17H12INO5

Notes

Research use only, not for human use.

Receptor

PI3K | IGF-1R

Available Sizes

Frequently Asked Questions

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