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GSK3368715 dihydrochloride

GSK3368715 dihydrochloride (EPZ019997 dihydrochloride) is an orally active and potent inhibitor of type I protein arginine methyltransferases (PRMTs), including PRMT1, PRMT3, PRMT4, PRMT6, and PRMT8. It exhibits anticancer and antitumor activity and can be used to study advanced solid tumors.

Product Specifications

CAS Number

1628925-77-8

Stability

≥ 2 years

Purity

>98% (HPLC)

Weight

439.46

Molecular Formula

C20H40Cl2N4O2

Notes

Research use only, not for human use.

Receptor

Histone Methyltransferase

Available Sizes

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