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Glutaminase-IN-1

Glutaminase-IN-1 (CB839 derivative), a novel 1,3,4-selenodiazepine inhibitor of the renal-type glutaminase (KGA) variant, exhibited antitumor activity in an aggressive H22 hepatocellular carcinoma xenograft model.

Product Specifications

CAS Number

2247127-79-1

Stability

≥ 2 years

Purity

>98% (HPLC)

Weight

618.47

Molecular Formula

C26H24F3N7O3Se

Notes

Research use only, not for human use.

Receptor

Transporter

Available Sizes

Curated Selection

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