GKI-1
GKI-1 is a Greatwall (GWL) kinase inhibitor with an IC50 of 4.9 for hGWLFL and 2.5 µM for hGWL-KinDom. It exhibits stronger inhibition on ROCK1 with an IC50 of 11 µM and only weakly inhibits PKA.
Product Specifications
CAS Number
2444764-03-6
Stability
≥ 2 years
Purity
>98% (HPLC)
Weight
269.73
Molecular Formula
C15H12ClN3
Notes
Research use only, not for human use.
Receptor
Others
Available Sizes
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