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DBPR112

DBPR112 is an orally active furanopyrimidine-based EGFR inhibitor with IC50s of 15 nM for EGFRWT and 48 nM for EGFRL858R/T790M, capable of occupying the ATP-binding site and demonstrating significant antitumor efficacy.

Product Specifications

CAS Number

1226549-49-0

Stability

≥ 2 years

Purity

>98% (HPLC)

Weight

533.62

Molecular Formula

C32H31N5O3

Notes

Research use only, not for human use.

Receptor

EGFR

Available Sizes

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