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CRA-026440 hydrochloride

CRA-026440 hydrochloride is a potent and broad-spectrum HDAC inhibitor. CRA-026440 hydrochloride exhibits Ki values against recombinant HDAC isoenzymes HDAC1, HDAC2, HDAC3, HDAC6, HDAC8, and HDAC10 are 4 nM, 14 nM, 11 nM, 15 nM, 7 nM, and 20 nM, respectively. CRA-026440 hydrochloride exhibits antitumor and antiangiogenic activities.

Product Specifications

CAS Number

847459-98-7

Stability

≥ 2 years

Purity

>98% (HPLC)

Weight

456.92

Molecular Formula

C23H25ClN4O4

Notes

Research use only, not for human use.

Receptor

HDAC

Available Sizes

Curated Selection

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