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BMS-470539 dihydrochloride

BMS-470539 dihydrochloride is a selective and highly potent melanocortin 1 receptor (MC-1 R) agonist with anti-inflammatory activity. BMS-470539 attenuates oxidative stress and neuronal apoptosis via the MC1R/cAMP/PKA/Nurr1 signaling pathway in a neonatal hypoxia-ischemia rat model.

Product Specifications

Stability

≥ 2 years

Purity

>98% (HPLC)

Weight

632.62

Molecular Formula

C32H43Cl2N5O4

Notes

Research use only, not for human use.

Receptor

Melanocortin Receptor

CAS Number

2341796-82-3

Available Sizes

Curated Selection

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