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Yangambin

Yangambin is a selective antagonist of the cardiovascular effects of platelet activating factor (PAF) ; it has hypotensive effect, which is probably due to a peripheral vasodilatation that involves, at least, the inhibition the Ca2+ influx through voltage-gated Ca2+ channels. Yangambin has central nervous system activity, it presents a depressant activity in the open field, forced swimming and pentobarbital sleeping time tests.

Product Specifications

CAS Number

13060-14-5

Stability

≥ 2 years

Purity

>98% (HPLC)

Weight

446.496

Molecular Formula

C24H30O8

Notes

Research use only, not for human use.

Receptor

Calcium Channel

Available Sizes

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