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TL-895

TL-895 is an ATP-competitive, and highly selective irreversible inhibitor of Bruton’s Tyrosine Kinase (BTK) . TL-895 showed good potency with an IC50 of 1.5 nM and a Ki of 11.9 nM.

Product Specifications

CAS Number

1415823-49-2

Stability

≥ 2 years

Purity

>98% (HPLC)

Weight

447.5

Molecular Formula

C25H26FN5O2

Notes

Research use only, not for human use.

Receptor

——

Available Sizes

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