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GSK778

GSK778 is a potent and selective inhibitor of BD1 bromodomain such as BRD2 BD1 (IC50s = 75 nM), BRD3 BD1 (IC50s = 41 nM), BRD4 BD1 (IC50s = 41 nM), and BRDT BD1 (IC50s = 143 nM) . GSK778 inhibits proliferation, induces a cell cycle arrest and apoptosis.

Product Specifications

CAS Number

2451862-42-1

Stability

≥ 2 years

Purity

>98% (HPLC)

Weight

511.61

Molecular Formula

C30H33N5O3

Notes

Research use only, not for human use.

Receptor

VHL

Available Sizes

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