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AZ12672857

AZ12672857 is an inhibitor of EphB4 with IC50 of 1.3 nM. AZ12672857 inhibits cell proliferation of Src transfected 3T3 cells with IC50 of 2 nM and autophosphorylation of EphB4 in transfected CHO-K1 cells with IC50 of 9 nM.

Product Specifications

CAS Number

945396-55-4

Stability

≥ 2 years

Purity

>98% (HPLC)

Weight

486.57

Molecular Formula

C26H30N8O2

Notes

Research use only, not for human use.

Receptor

——

Available Sizes

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