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Oritinib

Oritinib is an inhibitor of EGFR with IC50s of 18, 0.7, 4, 0.1, 1.4 and 0.89 nM for EGFR (wt), EGFR (L858R), EGFR (L861Q), EGFR (L858R/T790M), EGFR (d746-750), EGFR (d746-750/T790M), respectively. Oritinib can be used in studies about the treatment of non-small cell lung cancer.

Product Specifications

CAS Number

2035089-28-0

Stability

≥ 2 years

Purity

>98% (HPLC)

Weight

539.67

Molecular Formula

C31H37N7O2

Notes

Research use only, not for human use.

Receptor

——

Available Sizes

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