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YS-370

YS-370 is an orally active inhibitor of P-gp and shows moderate inhibition against CYP3A4. YS-370 effectively reverses multidrug resistance to paclitaxel and colchicine and exhibits stronger antitumor activity in combination with paclitaxel.

Product Specifications

CAS Number

2470908-79-1

Stability

≥ 2 years

Purity

>98% (HPLC)

Weight

663.6

Molecular Formula

C37H35BrN4O3

Notes

Research use only, not for human use.

Receptor

Enpp-1

Available Sizes

Curated Selection

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