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ARD-2128

ARD-2128 is a highly potent, orally bioavailable PROTAC androgen receptor (AR) degrader. ARD-2128 effectively reduces AR protein, suppresses AR-regulated genes in tumor tissues, and inhibits growth of tumor without signs of toxicity.

Product Specifications

CAS Number

2222111-87-5

Stability

≥ 2 years

Purity

>98% (HPLC)

Weight

820.38

Molecular Formula

C45H50ClN7O6

Notes

Research use only, not for human use.

Receptor

TNIK

Available Sizes

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