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CAY10781

CAY10781 is an inhibitor of the protein-protein interaction between neuropilin-1 (NRP-1) and VEGF-A.1It inhibits the interaction by 43% when used at a concentration of 12.5 μM. CAY10781 also inhibits VEGF-A-induced phosphorylation of VEGFR2 in catecholamine A-differentiated (CAD) cells when used at the same concentration.

Product Specifications

CAS Number

1210360-87-4

Stability

≥ 2 years

Purity

>98% (HPLC)

Weight

231.211

Molecular Formula

C11H9N3O3

Notes

Research use only, not for human use.

Receptor

Neutral sphingomyelinase

Available Sizes

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