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XY028-140

XY028-140 is a selective CDK4/CDK6 degrade and inhibits both CDK4/6 expression and activity in cancer cells. XY028-140 is a PROTAC connected by ligands for Cereblon and CDK.

Product Specifications

CAS Number

2229974-83-6

Stability

≥ 2 years

Purity

>98% (HPLC)

Weight

760.8

Molecular Formula

C39H40N10O7

Notes

Research use only, not for human use.

Receptor

Endogenous Metabolite|Apoptosis

Available Sizes

Curated Selection

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