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THZ1 2HCl

THZ1 2HCl is a selective, covalent, and allosteric inhibitor of CDK7 with an IC50 of 3.2 nM. THZ1 2HCl has antiproliferative effects on a variety of cancer cell lines.

Product Specifications

CAS Number

2095433-94-4

Stability

≥ 2 years

Purity

>98% (HPLC)

Weight

638.98

Molecular Formula

C31H30Cl3N7O2

Notes

Research use only, not for human use.

Receptor

CCR4

Available Sizes

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