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L-745870 trihydrochloride

L-745870 trihydrochloride is a highly potent and selective D4 dopamine receptor antagonist. L-745870 trihydrochloride exhibits moderate affinity for 5-HT2 receptors, sigma sites and α-adrenoceptors and shows weaker affinity for D2 and D3 receptors.

Product Specifications

CAS Number

866021-03-6

Stability

≥ 2 years

Purity

>98% (HPLC)

Weight

436.2

Molecular Formula

C18H22Cl4N4

Notes

Research use only, not for human use.

Receptor

Syk

Available Sizes

Curated Selection

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