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Org 25543 hydrochloride

Org 25543 hydrochloride is a potent and selective glycine transporter type 2 (GlyT2) inhibitor (IC50 = 16 nM for hGlyT2) . Displays no activity at GlyT1 or 56 other common biological targets (≥ 100 μM), in a glycine uptake assay in CHO cells.

Product Specifications

CAS Number

495076-64-7

Stability

≥ 2 years

Purity

>98% (HPLC)

Weight

448.99

Molecular Formula

C24H33ClN2O4

Notes

Research use only, not for human use.

Receptor

Antibacterial

Available Sizes

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