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K-756

K-756 is a direct and selective inhibitor of tankyrase (TNKS), which inhibits the ADP-ribosylation activity of TNKS1 (IC50 = 31 nM) and TNKS2 (IC50 = 36 nM) .

Product Specifications

CAS Number

130017-40-2

Stability

≥ 2 years

Purity

>98% (HPLC)

Weight

433.512

Molecular Formula

C24H27N5O3

Notes

Research use only, not for human use.

Receptor

URAT1

Available Sizes

Curated Selection

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