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ADAMTS-5 Inhibitor

ADAMTS-5 Inhibitor is a potent ADAMTS-5 (aggrecanase-2) inhibitor, with an IC50 of 1.1 μM. ADAMTS-5 Inhibitor shows >40-fold functional selectivity over ADAMTS-4 (aggrecanase-1) .

Product Specifications

Stability

≥ 2 years

Purity

>98% (HPLC)

Weight

449.91

Molecular Formula

C16H11ClF3N3OS3

Notes

Research use only, not for human use.

Receptor

5-HT2A| D1 receptor| D5 receptor

CAS Number

929634-33-3

Available Sizes

Curated Selection

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