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Sigma-1 receptor antagonist 3

Sigma-1 receptor antagonist 3 is a more potent and selective antagonist of Sigma-1 (σ1) receptor (Ki = 1.14 nM) than σ2 receptor (Ki = 1239 nM) .

Product Specifications

CAS Number

1639220-17-9

Stability

≥ 2 years

Purity

>98% (HPLC)

Weight

363.86

Molecular Formula

C19H23ClFN3O

Notes

Research use only, not for human use.

Receptor

——

Available Sizes

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