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EGFR-IN-5

EGFR-IN-5 is a selective inhibitor of EGFR. The IC50s for EGFR, EGFR (L858R), EGFR (L858R/T790M), and EGFR (L858R/T790M/C797S) are 10.4, 1.1, 34, 7.2 nM, respectively.

Product Specifications

CAS Number

2225887-26-1

Stability

≥ 2 years

Purity

>98% (HPLC)

Weight

571.705

Molecular Formula

C31H38FN9O

Notes

Research use only, not for human use.

Receptor

——

Available Sizes

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