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GS-143

GS143 is a selec­tive IκBα ubiquitination inhibitor with an IC50 of 5.2 μM for SCFβTrCP1-mediated IκBα ubiquitylation.

Product Specifications

CAS Number

916232-21-8

Stability

≥ 2 years

Purity

>98% (HPLC)

Weight

466.46

Molecular Formula

C28H19FN2O4

Notes

Research use only, not for human use.

Receptor

IκBα phosphorylation

Available Sizes

Curated Selection

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