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AS1810722

AS1810722 is an orally active and potent STAT6 inhibitor (IC50 :1.9 nM) . AS1810722 shows a good profile of CYP3A4 inhibition. AS1810722, a derivative of fused bicyclic pyrimidine, has the potential for allergic diseases such as asthma and atopic diseases research.

Product Specifications

CAS Number

909561-15-5

Stability

≥ 2 years

Purity

>98% (HPLC)

Weight

477.52

Molecular Formula

C25H25F2N7O

Notes

Research use only, not for human use.

Receptor

CYP3A4|STAT6

Available Sizes

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