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API-1

API-1 is a potent inhibitor of Akt. It induces GSK3-dependent, β-TrCP- and FBXW7-mediated Mcl-1 degradation, resulting in induction of apoptosis .

Product Specifications

CAS Number

36707-00-3

Stability

≥ 2 years

Purity

>98% (HPLC)

Weight

337.29

Molecular Formula

C13H15N5O6

Notes

Research use only, not for human use.

Receptor

Akt

Available Sizes

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