GSK046
GSK046 is a potent, selective and orally active BD2 bromodomain inhibitor of the BET proteins (IC50s of 264 nM (BRD2 BD2), 98 nM (BRD3 BD2), 49 nM (BRD4 BD2) and 214 nM (BRDT BD2), respectively) .
Product Specifications
CAS Number
2474876-09-8
Stability
≥ 2 years
Purity
>98% (HPLC)
Weight
414.48
Molecular Formula
C23H27FN2O4
Notes
Research use only, not for human use.
Receptor
BRD2-BD2|BRD3-BD2|BRD4-BD2|BRDT-BD2
Available Sizes
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