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NAcM-OPT HCl (2089293-61-6 free base)

NAcM-OPT HCL is an orally bioavailable cullin neddylation 1 (DCN1) inhibitor that targets N-Acetyl-UBE2M (E2 conjugating enzyme, UBC12) interaction with DCN1 with IC50 of 79 nM.

Product Specifications

CAS Number

2416146-10-4

Stability

≥ 2 years

Purity

>98% (HPLC)

Weight

470.86

Molecular Formula

C23H30Cl3N3O

Notes

Research use only, not for human use.

Receptor

DCN1-UBE2M

Available Sizes

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