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BDTX-189

BDTX-189 is a potent and selective inhibitor of allosteric EGFR and HER2 oncogenic mutations (KDs of 0.2, 0.76, 13 and 1.2 nM for EGFR, HER2, BLK and RIPK2, reapectively) . BDTX-189 exhibits anticancer activity.

Product Specifications

CAS Number

2414572-47-5

Stability

≥ 2 years

Purity

>98% (HPLC)

Weight

561.03

Molecular Formula

C29H29ClN6O4

Notes

Research use only, not for human use.

Receptor

BLK|EGFR|HER2|RIPK2

Available Sizes

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