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Bractoppin

Bractoppin is a drug-like inhibitor of phosphopeptide recognition by the human BRCA1 tandem (t) BRCT domain (IC50 = 0.074 μM), which selectively inhibits substrate binding with nanomolar potency in vitro.

Product Specifications

CAS Number

2290527-07-8

Stability

≥ 2 years

Purity

>98% (HPLC)

Weight

414.47

Molecular Formula

C25H23FN4O

Notes

Research use only, not for human use.

Receptor

Others

Available Sizes

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