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JAK/HDAC-IN-1

JAK/HDAC-IN-1 is an effective JAK2/HDAC dual inhibitor (IC50s: 4 and 2 nM for JAK2 and HDAC) . It also shows antiproliferative and proapoptotic activities in several hematological cell lines.

Product Specifications

CAS Number

2284621-75-4

Stability

≥ 2 years

Purity

>98% (HPLC)

Weight

450.32

Molecular Formula

C19H21Cl2N7O2

Notes

Research use only, not for human use.

Receptor

HDAC|HDAC2|HDAC6|HDAC8|JAK1|JAK2|JAK3|Tyk2

Available Sizes

Curated Selection

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